Ligustrazine Ligusticum chuanxiong ikuramo ibikoresho fatizo bya farumasi

Ibisobanuro bigufi:

Ligustrazine ni bioactive igizwe na Ligusticum chuanxiong, imiti gakondo ikoreshwa mubushinwa.Irashobora kubuza gukusanya platine, kongera vasodilasiya, kongera amaraso yubwonko kandi ikagira ingaruka za neuroprotective.Gutera Ligustrazine byakoreshejwe cyane mu kuvura indwara ziterwa na ischemic stroke, indwara z'umutima, indwara ya diabete ya nepropatique na osteoarthritis yo mu ivi mu Bushinwa.Ligustrazine yasuzumwe kandi nk'ubuvuzi bwo kuvura ibisebe by'umuvuduko, nk'umuti wo gukiza abarwayi bafite lymphoma itari Hodgkin, ndetse nk'ubuvuzi bwa asima ya bronchial na vertebrobasilar idahagije.


Ibicuruzwa birambuye

Ibicuruzwa

Amakuru y'ibicuruzwa

Ligustrazine ni bioactive igizwe na Ligusticum chuanxiong, imiti gakondo ikoreshwa mubushinwa.Irashobora kubuza gukusanya platine, kongera vasodilasiya, kongera amaraso yubwonko kandi ikagira ingaruka za neuroprotective.Gutera Ligustrazine byakoreshejwe cyane mu kuvura indwara ziterwa na ischemic stroke, indwara z'umutima, indwara ya diabete ya nepropatique na osteoarthritis yo mu ivi mu Bushinwa.Ligustrazine yasuzumwe kandi nk'ubuvuzi bwo kuvura ibisebe by'umuvuduko, nk'umuti wo gukiza abarwayi bafite lymphoma itari Hodgkin, ndetse nk'ubuvuzi bwa asima ya bronchial na vertebrobasilar idahagije.
1 、 Ibiranga Ligustrazine
Ligustrazine ni kirisiti ya acicular itagira ibara ifite aho ishonga ya 80-82 ° (kugena microscopique) hamwe no guteka kwa 190 °.Ifite impumuro idasanzwe, hygroscopicity na sublimation yoroshye.Irashobora gushonga byoroshye mumazi ashyushye hamwe na peteroli ya ether, chloroform hamwe na acide hydrochloric, gushonga gato muri ether kandi ntigashonga mumazi akonje.
2 、 Ingaruka za Ligustrazine
1. Ingaruka ku mutima
2. Ongera imitsi ya koronari
3. Kugura imiyoboro y'amaraso ya peripheri no kugabanya umuvuduko w'amaraso
4. Kunoza ubwonko bwubwonko
5. Kubuza gukusanya platine na antithrombotic
6. Ingaruka kuri sisitemu yinkari
7. Kunoza microcrolluction
8. Ingaruka kuri sisitemu y'ubuhumekero
9. Kurwanya ikibyimba
10. Kongera imikorere yubudahangarwa
11. Kurwanya imishwarara no gukangurira imirasire
3 mode Uburyo bwo gukora bwa Ligustrazine
Dimethylpyrazine yateguwe no guhuza butanone hamwe na nitrite ya Ethyl kugirango itange dimethylglyoxime, hanyuma igabanywa kandi irazunguruka.Ibicuruzwa byizunguruka byerekanwa na parike, hanyuma distillate ikonjeshwa, ikabikwa kandi ikayungurura kugirango ibone ibicuruzwa bya tetramethylpyrazine.Gusubiramo amazi hamwe na carbone decolorisation ikoreshwa mugutunganya.Mugihe utegura hydrochloride, umuti wa Ethanol urimo 15% - 20% hydrogène chloride irashobora kongerwaho ibitonyanga kuri acetone kugirango ibe umunyu
4 field Imirima ikoreshwa ya Ligustrazine
1. Inganda zimiti: kubyara ibiyobyabwenge.
2. Inganda zibiribwa: zikoreshwa nkibintu biryoha, byongera ibinyobwa bisindisha, uburyohe hamwe ninyongera y itabi.

Ibipimo byibicuruzwa

UMWUGA W'ISHYAKA
izina RY'IGICURUZWA ligustrazine
CAS 1124-11-4
Imiti yimiti C8H12N2
Brand Hande
Muruganda Yunnan Hande Bio-Tech Co, Ltd.
Country Kunming,China
Hashyizweho 1993
 BAMAKURU ASIC
Synonyme Tetramethylpyrazine; 2,3,5,6-tetramethylpyrazine;Pyrazine, tetramethyl-;
Imiterere  24
Ibiro 136.19400
HS Kode N / A.
UbwizaSpecification Ibisobanuro bya sosiyete
Certificates N / A.
Suzuma Guhitamo ukurikije ibyo abakiriya bakeneye
Kugaragara Kirisiti idafite amabara
Uburyo bwo gukuramo rhizome ya chuanxiong
Ubushobozi bwa buri mwaka Guhitamo ukurikije ibyo abakiriya bakeneye
Amapaki Guhitamo ukurikije ibyo abakiriya bakeneye
Uburyo bwo Kwipimisha N / A.
Ibikoresho Kugwizaubwikorezis
PaymentTerms T / T, D / P, D / A.
Other Emera ubugenzuzi bwabakiriya igihe cyose;Fasha abakiriya kwiyandikisha kugenga.

 

Tanga ibicuruzwa

1.Ibicuruzwa byose byagurishijwe nisosiyete ni ibikoresho byarangije igice.Ibicuruzwa byibanda cyane cyane kubabikora bafite ibyangombwa byo gukora, kandi ibikoresho fatizo ntabwo aribicuruzwa byanyuma.
2.Ibishobora kuba byiza nibisabwa mugutangiza byose biva mubitabo byatangajwe.Umuntu ku giti cye ntabwo asaba gukoresha mu buryo butaziguye, kandi kugura kugiti cye byanze.
3.Amashusho nibicuruzwa byamakuru kururu rubuga bireba gusa, kandi ibicuruzwa nyirizina bizatsinda.


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