Amakuru y'ibicuruzwa
Artesunate ikozwe mubintu byiza artemisinin yakuwe muri Artemisia annua, idasanzwe mubushinwa, ikoresheje synthesis.Cyakora cyane cyane kuri clone yicyiciro gitukura cya malariya.Nibintu byonyine bikomoka kuri artemisinin ishobora gukorwa mubikorwa byogushonga amazi muri iki gihe.Irashobora kwica Plasmodium mugice cya erythrocytike kandi ikagera kuri antimalarial.Ifite ibiranga ibikorwa byinshi bya antimalariya, antipyretike yihuse, igihe gito cyo guhindura nabi Plasmodium, hamwe nuburozi buto ningaruka mbi.Nibwo buryo bwa mbere bwo kuvura malariya ikabije.
1 inkomoko y'ibihingwa
Artesunate nigice cya sintetike ya artesunate ikomoka.
2 ism Uburyo bwibikorwa
Uburyo bwibikorwa bya artesunate artemisinin.Irabanza ikora ku biryo bya viticle membrane, hejuru yubutaka na mitochondriya ya Plasmodium.Iya kabiri ni membrane membrane na retopulum ya endoplasme.Mubyongeyeho, igira kandi ingaruka runaka kuri chromatine muri nucleus.Nkuko iki gicuruzwa kibanza gukora kuri membrane bubble membrane, bityo bikabuza gufata intungamubiri, parasite ya malariya ihita yicwa ninzara ya acide amine, ikora vuba imitsi ya autophagic, kandi igakomeza gusohoka mumubiri, igatakaza cytoplazme nyinshi hanyuma igapfa.
Uruhare
1. Imiti igabanya ubukana
Artesunate ni imiti ikoreshwa cyane.Nibikomoka kuri artesunate hamwe na sesquiterpene lactone yubatswe, ikaba yagabanijwe artesunate.
2. Ingaruka zishobora kurwanya antikanseri
Artesunate igira ingaruka zikomeye zo kwica kanseri yibibyimba kandi ntabwo byoroshye kubyara imiti.Mu myaka yashize, intiti zo mu gihugu ndetse no mu mahanga zabonye ko artesunate ishobora kugira uruhare mu kurwanya ibibyimba mu gukumira ikwirakwizwa ry’uturemangingo tw’ibibyimba, gutera gutandukanya uturemangingo tw’ibibyimba na apoptose, kugenzura kwanduza ibimenyetso by’ingirabuzimafatizo, kubuza ibibyimba angiogenezi, kubuza gutera ibibyimba na metastasis, gukangurira anti -tumor imiti ya chimiotherapie no guhindura imiti irwanya.
4 field Umwanya wo gusaba
1. Inganda zimiti
Ibipimo byibicuruzwa
UMWUGA W'ISHYAKA | |
izina RY'IGICURUZWA | Artesunate |
CAS | 88495-63-0 |
Imiti yimiti | C19H28O8 |
Brand | Hande |
Muruganda | Yunnan Hande Bio-Tech Co, Ltd. |
Country | Kunming,China |
Hashyizweho | 1993 |
BAMAKURU ASIC | |
Synonyme | ARTENSUNATE; Butanedioicacid, 1 - ] -1,2-benzodioxepin-10-yl] ester; Artesunate (3R, 5aS, 6R, 8aS, 9R, 10S, 12R, 12aR) -Decahydro-3,6,9-trimethyl-3,12-epoxy-12H -pyrano (4,3-j) -Igitabo cya Himiki1,2-benzodioxepin-10-olhydrogensuccinate; ARTESUNATE; ArtesunateC19H28O8; Artemisininmonosuccine; , 6,9-trimethyl-3,12-epoxy-12H-pyrano [4,3-j] -1,2-benzodioxepin-10-yl] Ester |
Imiterere | |
Ibiro | 384.42 |
HS Kode | N / A. |
UbwizaSpecification | Ibisobanuro bya sosiyete |
Certificates | N / A. |
Suzuma | Guhitamo ukurikije ibyo abakiriya bakeneye |
Kugaragara | Kirisiti yera |
Uburyo bwo gukuramo | Artemisia annua Linn. |
Ubushobozi bwa buri mwaka | Guhitamo ukurikije ibyo abakiriya bakeneye |
Amapaki | Guhitamo ukurikije ibyo abakiriya bakeneye |
Uburyo bwo Kwipimisha | HPLC |
Ibikoresho | Kugwizaubwikorezis |
PaymentTerms | T / T, D / P, D / A. |
Other | Emera ubugenzuzi bwabakiriya igihe cyose;Fasha abakiriya kwiyandikisha kugenga. |
Tanga ibicuruzwa
1.Ibicuruzwa byose byagurishijwe nisosiyete ni ibikoresho byarangije igice.Ibicuruzwa byibanda cyane cyane kubabikora bafite ibyangombwa byo gukora, kandi ibikoresho fatizo ntabwo aribicuruzwa byanyuma.
2.Ibishobora kuba byiza nibisabwa mugutangiza byose biva mubitabo byatangajwe.Umuntu ku giti cye ntabwo asaba gukoresha mu buryo butaziguye, kandi kugura kugiti cye byanze.
3.Amashusho nibicuruzwa byamakuru kururu rubuga bireba gusa, kandi ibicuruzwa nyirizina bizatsinda.
Uruganda:
Yunnan hande Biotechnology Co., Ltd., yashinzwe muri Kanama 1993, ni uruganda rukora ubuhanga buhanitse mu bushakashatsi no guteza imbere ibinyabuzima.Nyuma yimyaka yiterambere, hande yashyizeho sisitemu nziza yubuziranenge, igenzura ubuziranenge bwibicuruzwa ukurikije ibipimo bihanitse, kandi byongera agaciro k’umusaruro wubushobozi.Ibicuruzwa byayo byatsinze icyemezo cy’amategeko n'amabwiriza mpuzamahanga, kandi gihinduka uruganda rukora ibikoresho bibisi bituma buri wese yumva yisanzuye.
Ba umutanga mwiza wibikoresho fatizo ninganda zifite ubunyangamugayo!
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