Amakuru y'ibicuruzwa
Dihydroartemisinin ni inkomoko ya artemisinin, igira ingaruka zikomeye kandi zihuse ku bwicanyi bwa erythrocytike ya parasite ya malariya, kandi irashobora kugenzura vuba ibitero by’amavuriro n'ibimenyetso.
1 plant Igiterwa gikomoka
Dihydroartemisinin ikomoka kuri artemisinin.Artemisinin ni imiti igabanya ubukana yakuwe muri Artemisia annua.
Uruhare
Igikorwa cya farumasi ya dihydroartemisinin gisa na artemisinin.Ingaruka ya artemisinin kuri ultrastructure ya Plasmodium falciparum mugice cya erythrocytique ni uguhindura imiterere ya membrane.Uyu muti ubanza ukora ibiryo byitwa viticle membrane, membrane membrane na mitochondria, bigakurikirwa na membrane nucleaire na reticulum ya endoplasme.Mubyongeyeho, binagira ingaruka kuri chromatine muri nucleus.Irashobora gukora kuri membrane vitamine ibiryo, ikabuza icyiciro cyambere cyo gufata imirire ya parasite ya malariya, bigatuma malariya ya malariya yicwa ninzara ya acide amine, igahita ikora vitamine autophagic, kandi igakomeza gusohoka mumubiri, igatakaza umubare munini cytoplazme nintungamubiri, ariko ntizuzuzwe, nuko ipfa vuba.Uburyo bwibikorwa byabwo ahanini ni ukubangamira imikorere ya Plasmodium surface membrane mitochondria.Binyuze mu kiraro cyacyo cya peroxide (dioxyde), cyahujwe nicyuma cyubusa cyakozwe nyuma yo kubora kwa hemoglobine kugirango habeho radicals yubusa idahindagurika hamwe na / cyangwa nabandi bahuza amashanyarazi, hanyuma igakora inyongeramusaruro hamwe na proteyine za parasite ya malariya, bikavamo urupfu rwa malariya.Kwakira tritium yanditseho isoleucine na Plasmodium falciparum yumuco muri vitro nayo yerekanye ko uburyo bwambere bwibikorwa bishobora kuba uguhagarika synthesis ya proteine ya Plasmodium.
3 field Umwanya wo gusaba
1. Inganda zimiti
Ibipimo byibicuruzwa
UMWUGA W'ISHYAKA | |
izina RY'IGICURUZWA | Dihydroartemisinin |
CAS | 81496-82-4 |
Imiti yimiti | C15H24O5 |
Brand | Hande |
Muruganda | Yunnan Hande Bio-Tech Co, Ltd. |
Country | Kunming,China |
Hashyizweho | 1993 |
BAMAKURU ASIC | |
Synonyme | . (3R, 5aS, 6R, 8aS, 9R, 12S, 12aR) (3H) inzoga; Dihydroartemisinin; Dihxdroarteannui; Dihydroartemisinin USP / EP / BP |
Imiterere | |
Ibiro | 284.35 |
HS Kode | N / A. |
UbwizaSpecification | Ibisobanuro bya sosiyete |
Certificates | N / A. |
Suzuma | Guhitamo ukurikije ibyo abakiriya bakeneye |
Kugaragara | Kirisiti yera |
Uburyo bwo gukuramo | Artemisia annua Linn. |
Ubushobozi bwa buri mwaka | Guhitamo ukurikije ibyo abakiriya bakeneye |
Amapaki | Guhitamo ukurikije ibyo abakiriya bakeneye |
Uburyo bwo Kwipimisha | HPLC |
Ibikoresho | Kugwizaubwikorezis |
PaymentTerms | T / T, D / P, D / A. |
Other | Emera ubugenzuzi bwabakiriya igihe cyose;Fasha abakiriya kwiyandikisha kugenga. |
Tanga ibicuruzwa
1.Ibicuruzwa byose byagurishijwe nisosiyete ni ibikoresho byarangije igice.Ibicuruzwa byibanda cyane cyane kubabikora bafite ibyangombwa byo gukora, kandi ibikoresho fatizo ntabwo aribicuruzwa byanyuma.
2.Ibishobora kuba byiza nibisabwa mugutangiza byose biva mubitabo byatangajwe.Umuntu ku giti cye ntabwo asaba gukoresha mu buryo butaziguye, kandi kugura kugiti cye byanze.
3.Amashusho nibicuruzwa byamakuru kururu rubuga bireba gusa, kandi ibicuruzwa nyirizina bizatsinda.